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Updated: Jul 12, 2025

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在实验室中对通用禁令规避的化合成大麻素受体激活剂及其类似物进行大麻素活性分析

Marie H Deventer1, Mattias Persson2, Caitlyn Norman3

  • 1Laboratory of Toxicology, Department of Bioanalysis, Faculty of Pharmaceutical Sciences, Ghent University, Ghent, Belgium.

Drug testing and analysis
|October 30, 2023
PubMed
概括

新的合成大麻素,包括没有尾巴的ADB-5'Br-INACA和MDMB-5'Br-INACA,保留了大麻素受体 (CB) 活性. 去除减少了CB1活性,而替代增加了CB1和CB2受体的强度和有效性.

关键词:
在ADB-5Br-BUTINACAA中在ADB-5Br-INACAA中.CB1类大麻素受体 CB1类大麻素受体在MDMB-5Br-INACAA中.化合成大麻素受体激活剂 化合成大麻素受体激活剂

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