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Updated: Jul 11, 2025

Microwave-Assisted Preparation of 1-Aryl-1H-pyrazole-5-amines
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对抗中性友性炎症的皮拉衍生物的设计和合成

Ko-Hua Yu1, Kai-Wen Tien2, Wei-Chun Wang1

  • 1School of Pharmacy, College of Medicine, National Cheng Kung University, Tainan, 701, Taiwan.

European journal of medicinal chemistry
|November 2, 2023
PubMed
概括

研究人员开发了新的固酶4 (PDE4) 抑制剂,通过向中性粒细胞来减少炎症. 化合物58和59强烈抑制了超氧化离子生成,为新的抗炎药物提供了潜力.

关键词:
作为一个中性粒细胞.这是一种超氧化离子.在YC-1中,YC-1是YC-1.

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