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Updated: Jul 11, 2025

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作为芳香酶抑制剂的 triazole 类似物的设计和药理学研究

Laxmi Banjare1,2

  • 1School of Pharmaceutical Sciences, Guru Ghasidas Central University, Bilaspur, 495009 (C.G.) India.

Anti-cancer agents in medicinal chemistry
|November 3, 2023
PubMed
概括

研究人员设计了100种新的三醇类似物作为芳香酶抑制剂,用于对抗乳腺癌. 化合物01表现出强烈的活性,显示出开发有毒性降低的向治疗的前景.

关键词:
3D-QSAR 是一个3D-QSAR.芳香酶抑制剂的使用芳香的味道让人感到愉快.乳腺癌 乳腺癌 乳腺癌莱特罗斯 (Letrozole) 是一种三醇类似物.三醇类似物.

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