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Updated: Jul 10, 2025

Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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通过Zincke中间体对皮里丁的区域分离化

Haiwen Wang1, Michael F Greaney1

  • 1School of Chemistry, The University of Manchester, Oxford Road, Manchester, M13 9PL, UK.

Angewandte Chemie (International ed. in English)
|November 20, 2023
PubMed
概括

这项研究引入了一种新型的pyridines的 arylation方法,使用一个环开通的Zincke中间体. 这种方法可以实现区域选择性催化或无金属的化,为二基提供了一条通往二的多功能途径.

关键词:
催化剂是一种催化剂.C−H 激活方式帕拉是什么意思?帕拉是什么意思?氨酸是什么? 氨酸是什么?

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