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Updated: Jul 10, 2025

Quantitative Structure-Activity Relationship, Activity Prediction, and Molecular Dynamics of Non-nucleotide Reverse Transcriptase Inhibitors
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设计,合成,对接研究和生物评估的新的2-Hydroxyacetophenone衍生物作为抗HIV-1的代理商

Samira Sooreni Oliaie1, Mahdieh Safakish1, Rouhollah Vahabpour Roudsari2

  • 1Department of Pharmaceutical Chemistry, School of Pharmacy, Shahid Beheshti University of Medical Sciences, Tehran, Iran.

Current HIV research
|November 22, 2023
PubMed
概括

研究人员开发了基于HIV整合酶抑制剂药的新型抗HIV-1药剂. 合成的化合物显示中度活性和低细胞毒性,为新药开发提供了有希望的基础.

关键词:
2-氧乙烯二氧化烯.设计设计设计设计设计设计.停靠对接 停靠对接艾滋病毒-1.艾滋病毒-1.整合酶可以整合.综合合成 综合合成

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