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Updated: Jul 10, 2025

Facile Preparation of 4-Substituted Quinazoline Derivatives
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Facile Preparation of 4-Substituted Quinazoline Derivatives

Published on: February 15, 2016

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使用L-proline作为催化剂的4-Aryl-4,9-dihydro-1H-pyrazolo[3,4-b]quinolines的多元组分合成-它真的可以进行吗?

Andrzej Danel1, Elżbieta Porębska1, Kacper Markiel1

  • 1The Faculty of Materials Engineering and Physics, Krakow University of Technology, Podchorążych Street 1, 30-084 Krakow, Poland.

Molecules (Basel, Switzerland)
|November 25, 2023
PubMed
概括

研究人员寻求一种新的合成pyrazoloquinolines,但发现报告的方法实际上产生了bis(pyrazol-5-oles). 这项研究纠正了这些重要异环化合物的有缺陷的合成程序.

关键词:
4,4-(甲基) -bis- ((3-甲基-1-甲基醇-5-) -oles) 的使用情况.4-阿里-4,9H-3-甲基-1--1-H-pyrazolo [3,4-b] 氨基.对于L-proline来说,这是一个很好的方法.多组分反应是多组分反应.

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