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Updated: Jul 9, 2025

Protocol for the Synthesis of Ortho-trifluoromethoxylated Aniline Derivatives
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Protocol for the Synthesis of Ortho-trifluoromethoxylated Aniline Derivatives

Published on: January 19, 2016

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铜介导的N-三甲基化O-基氧胺的N-三甲基化

Thomas D Fleetwood1,2, William J Kerr2, Joseph Mason1

  • 1Medicinal Chemistry, GSK Medicines Research Centre, Gunnels Wood Road, SG1 2NY, Stevenage, England, U.K.

Chemistry (Weinheim an der Bergstrasse, Germany)
|November 29, 2023
PubMed
概括

开发了一种用于二次胺的N-trifluoromethylation的新方法. 这种铜催化方法提供了一种简单,温和和经济有效的方法来合成新型N-CF3化合物.

关键词:
氨基化是指氨基化.催化剂是一种催化剂.铜铜 铜铜 铜铜N-三甲基亚胺是三甲基亚胺的一种.三甲基三化物.

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