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Updated: Jul 9, 2025

Microwave-Assisted Preparation of 1-Aryl-1H-pyrazole-5-amines
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Published on: June 23, 2019

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合成和矢量函数化pyrazolo[3,4-c]pyridines的合成和矢量函数化

Elizabeth V Bedwell1, Flavio da Silva Emery2, Giuliano C Clososki2

  • 1Department of Chemistry, University of Durham South Road Durham DH1 3LE UK p.g.steel@durham.ac.uk.

RSC advances
|November 29, 2023
PubMed
概括

研究人员合成了新的5-halo-1H-pyrazolo[3,4-c]pyridine支架,用于基于碎片的药物发现 (FBDD). 这些多功能异环化合物可以在多个位置选择性地功能化,从而实现高效的优化.

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