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Updated: Jul 9, 2025

A Platform of Anti-biofilm Assays Suited to the Exploration of Natural Compound Libraries
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Published on: December 27, 2016

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青素结合蛋白 (PBP) 抑制剂的开发:一个10年的化学前景

Ariane F Bertonha1, Caio C L Silva1, Karina T Shirakawa1,2

  • 1Brazilian Biosciences National Laboratory (LNBio), CNPEM, Campinas 13084-971, Brazil.

Experimental biology and medicine (Maywood, N.J.)
|November 29, 2023
PubMed
概括

新的研究探索了向细菌青素结合蛋白 (PBPs) 的抑制剂,以对抗抗生素耐药性. 本综述侧重于通过检查PBP转酶域抑制剂及其结构-活性关系来开发新型抗菌剂.

关键词:
青素结合蛋白是一种青素结合蛋白.抑制剂 抑制剂 抑制剂其他非β-乳糖抑制剂.基板类型的类似物.在β-lactams中使用.

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