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Updated: Jun 14, 2026

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors

Published on: October 26, 2015

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拼接类作为潜在的细胞透性抑制剂的致癌性DAXX蛋白DAXX蛋白

Clare Jelinska1,2,3, Srinivasaraghavan Kannan4, Yuri Frosi5

  • 1NTU Institute of Structural Biology, Experimental Medicine Building Level 06-01, 59 Nanyang Drive 636921 Singapore csiclar@nus.edu.sg.

RSC chemical biology
|November 30, 2023
PubMed
概括

研究人员开发了针对DAXX (死亡域关联蛋白6),一种在癌症中高调的蛋白质的新型合. 这些抑制DAXX,扰乱癌症的进展,并显示治疗潜力.

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