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小分子CD73抑制剂:最近的进展和未来的前景.

Gong-Hui Ge1, Qiu-Yin Wang1, Zhen-Hao Zhang1

  • 1School of Pharmacy / Key Laboratory of Research and Development of Small Molecule Targeted Antitumor Drugs, China Medical University, 77 Puhe Road, North New Area, Shenyang 110122, China.

European journal of medicinal chemistry
|December 12, 2023
PubMed
概括

抑制CD73是一种对瘤生长和转移至关重要的酶,可以减少腺介导免疫抑制. 这种方法为开发针对固体瘤的新型小分子抗瘤药物提供了有前途的战略.

关键词:
亚丁氨酸 (Adenosine) 是一种氨基酸.CD73 CD73 CD73 CD73 CD73 CD73 CD73 CD73 CD73 CD73结构与活动的关系.

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