对潜在的CDC7激酶抑制剂的结构和在中的研究

Mohanbabu Mookkan1, Saravanan Kandasamy2, Abdel-Basit Al-Odayni3

  • 1Department of Physics, Presidency College (Autonomous), University of Madras, Chennai 600 005, India.

ACS omega
|December 18, 2023
PubMed
概括

合成和表征了两种新型的pyrazole衍生物,即PYRA-1和PYRA-2. 分子模拟表明PYRA-2是CDC7激酶的更强大的抑制剂,这是潜在的癌症治疗标.