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Updated: Jul 7, 2025

Parallel Interrogation of β-Arrestin2 Recruitment for Ligand Screening on a GPCR-Wide Scale using PRESTO-Tango Assay
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Published on: March 10, 2020

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孤儿受体GPR101与逮捕因的基础相互作用导致了构成性内化

Dayana Abboud1, Clauda Abboud1, Asuka Inoue2

  • 1Laboratory of Molecular Pharmacology, GIGA-Molecular Biology of Diseases, University of Liege, Liege, Belgium.

Biochemical pharmacology
|December 27, 2023
PubMed
概括

G蛋白结合受体101 (GPR101) 与逮捕因相互作用,导致其内部化和降解. 这种构成性贩运调节GPR101信号,影响生长激素分泌和X链接巨症候群 (X-LAG).

关键词:
在被捕后,我被捕了.克拉特林 (Clathrin) 是一个名为克拉特林的词汇.构成性活动 构成性活动在 GPR101 中,GPR101 是一个简单的语法.内部化 内部化 内部化孤儿的GPCRR是一个孤儿.

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