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Updated: Jul 5, 2025

A Two-Step Protocol for Umpolung Functionalization of Ketones Via Enolonium Species
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A Two-Step Protocol for Umpolung Functionalization of Ketones Via Enolonium Species

Published on: August 16, 2018

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可见光促进的α-C ((sp3) -H氨基化以与醇和胺

Yaqi Deng1, Zongjing Hu1, Jian Xue1

  • 1Shanghai Engineering Research Center of Molecular Therapeutics and New Drug Development, East China Normal University, Shanghai 200062 China.

Organic letters
|January 19, 2024
PubMed
概括

一个新的可见光驱动反应使使用胺和醇的乙烯有效的C-H氨基化成为可能. 该方法采用2,3-二-5,6-二-p-基 (DDQ) 和三丁酸盐 (TBN),为骨髓瘤药物发现产生有前途的化合物.

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