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Updated: Jul 4, 2025

A Simple Bioassay for the Evaluation of Vascular Endothelial Growth Factors
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关于VEGFR2氨酸激酶抑制剂的结构-活性关系研究,用于识别潜在的天然抗癌化合物

Meenakshi Verma1,2, Aqib Sarfraz3, Inamul Hasan3

  • 1Plant Biotechnology Division, CSIR-Central Institute of Medicinal and Aromatic Plants, P.O.- CIMAP, Kukrail Picnic Spot Road, Lucknow 226015 (Uttar Pradesh), India.

Medicinal chemistry (Shariqah (United Arab Emirates))
|February 1, 2024
PubMed
概括

这项研究开发了一种定量结构-活性关系 (QSAR) 模型,以确定天然化合物作为潜在的VEGFR2抑制剂. 一些天然化合物,包括Lavendustin_A,显示出有前途的抑制活性和结合亲和力,为现有药物提供了替代品.

关键词:
接收人 接收人在QSAR中使用QSAR.在VEGFR2的基础上,VEGFR2动力学模拟的动力学模拟抑制剂. 抑制剂. 这些分子对接的分子对接.铁氨酸激酶酶的使用方法

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