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Updated: Jul 4, 2025

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检测和描述GPER结合部位:基于黄胺的对接和分子动力学模拟研究.

David Méndez-Luna1, Sonia Guzmán-Velázquez2, Itzia-Irene Padilla-Martínez3

  • 1Laboratorio de Diseño y Desarrollo de Nuevos Fármacos e Innovación Biotecnológica, Escuela Superior de Medicina, Instituto Politécnico Nacional, Plan de San Luis y Díaz Mirón s/n, Col. Casco de Santo Tomas, Alcaldía Miguel Hidalgo, C.P. 11340 Ciudad de México, Mexico; Departamento de Fisiología, Escuela Nacional de Ciencias Biológicas, Instituto Politécnico Nacional, Zacatenco, Av. Wilfrido Massieu 399, Col. Nueva Industrial Vallejo, Alcaldía Gustavo A. Madero, C.P. 07738 Ciudad de México, Mexico.

The Journal of steroid biochemistry and molecular biology
|February 2, 2024
PubMed
概括

黄类药物通过与G蛋白结合雌激素受体 (GPER) 相互作用,显示出作为辅助癌症治疗的前景. 像普埃拉林这样的特定黄类药物可能会调节GPER,提供潜在的抗癌作用.

关键词:
有约束力的网站停靠对接 停靠对接黄类化合物 黄类化合物一个GPER的医生.分子动力学模拟的模拟.

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