使

Tao Liu1, Zejun Peng1, Manting Lai1

  • 1Affiliated Cancer Hospital, Guangdong Provincial Key Laboratory of Molecular Target & Clinical Pharmacology, School of Pharmaceutical Sciences, Guangzhou Medical University, No.1 Xinzao, Panyu District, Guangzhou 511436, China.

概括

一种新型的 ynamide 合试剂能够使用未受保护的氨基酸进行反向合成,克服了 60 年的挑战. 这种具有成本效益的绿色化学方法有助于有效制造治疗性.