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Updated: Jul 6, 2026

Regioselective O-Glycosylation of Nucleosides via the Temporary 2',3'-Diol Protection by a Boronic Ester for the Synthesis of Disaccharide Nucleosides
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使用基于时间解析的寡核酸的药物查平台,重新将固糖酸作为抗前列腺癌的 uracil DNA glycosylase 抑制剂

Sang-Cuo Nao1, Le-Sheng Huang1, Daniel Shiu-Hin Chan2

  • 1State Key Laboratory of Quality Research in Chinese Medicine, Institute of Chinese Medical Sciences, University of Macau, Taipa, Macau 999078, China.

Bioorganic chemistry
|February 8, 2024
PubMed
概括

药物重定向通过时间解析光谱加速,克服了高通量查中的光问题. 固醇被确定为 uracil-DNA glycosylase (UDG) 的强有力的抑制剂,显示出癌症治疗的前景.

关键词:
药物重新定位是药物重新定位.药物查是指对药物进行查.(III) 复合物 (III) 复合物时间解析的排放量.乌拉-DNA葡萄糖酶是什么

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