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Updated: Jul 4, 2025

Facile Preparation of 4-Substituted Quinazoline Derivatives
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Facile Preparation of 4-Substituted Quinazoline Derivatives

Published on: February 15, 2016

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新的阿尔法9nAChR联体 基于一个5-(昆利丁-3-ylmethyl) -1,2,4-oxadiazole 基架

Clelia Dallanoce1, Katrin Richter2, Clare Stokes3

  • 1Department of Pharmaceutical Sciences, Medicinal Chemistry Section "Pietro Pratesi″, University of Milan, Via L. Mangiagalli 25, 20133 Milan, Italy.

ACS chemical neuroscience
|February 9, 2024
PubMed
概括

研究人员确定了新的向尼古丁乙胆受体 (nAChR) 的化合物,其中包含α9亚单元. 这些分子,QMO-28 (激动剂) 和QMO-17 (对抗剂),显示了通过胆固醇抗炎系统 (CAS) 管理炎症性疼痛的潜力.

关键词:
药物开发是药物的发展.听到 听到 听到 听到 听到 听到 听到这是一种炎症炎症炎症炎症.尼古丁酸尼古丁酸的使用方法药理学 药理学 药理学 药理学 药理学电压的压力.

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