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Updated: Jul 3, 2025

Parallel Interrogation of β-Arrestin2 Recruitment for Ligand Screening on a GPCR-Wide Scale using PRESTO-Tango Assay
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Parallel Interrogation of β-Arrestin2 Recruitment for Ligand Screening on a GPCR-Wide Scale using PRESTO-Tango Assay

Published on: March 10, 2020

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GPCR树的黑暗面 - - 对未被充分研究的GPCR的研究进展

Magdalena M Scharf1, Laura J Humphrys2, Sandra Berndt3

  • 1Karolinska Institutet, Dept. Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Stockholm, Sweden.

British journal of pharmacology
|February 10, 2024
PubMed
概括

许多研究不足的G蛋白结合受体 (GPCR) 具有尚未开发的治疗潜力. 本综述探讨了研究这些重要受体的知识差距和策略,包括嗅觉和味觉受体.

关键词:
有毛的动物.与G蛋白结合的受体是G蛋白结合的受体.附着性 GPCRs 的附着性嗅觉受体是一种嗅觉受体.孤儿受体是一种孤儿受体.味道受体的味道受体.没有研究过的GPCR.

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