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Updated: Jul 3, 2025

Protocol for the Synthesis of Ortho-trifluoromethoxylated Aniline Derivatives
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Protocol for the Synthesis of Ortho-trifluoromethoxylated Aniline Derivatives

Published on: January 19, 2016

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一种SmI2介导的减少循环反应,使用三乙胺组作为激素前体

Kota Yoshioka1, Hiroki Iwasaki1, Mako Hanaki1

  • 1Kyoto Pharmaceutical University, 1 Misasagi-Shichono-cho, Yamashina-ku, Kyoto, 607-8412, Japan. iwasaki@mb.kyoto-phu.ac.jp.

Organic & biomolecular chemistry
|February 16, 2024
PubMed
概括

研究人员开发了一种新型的三介导的还原循环化方法,用于从具有挑战性的非循环胺基前体中合成2 - 三甲林多林. 该方法还可以将其转化为2-trifluoromethylindoles.

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Radical Reactivity: Intramolecular vs Intermolecular

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