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Updated: Jul 2, 2025

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
07:16

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission

Published on: August 16, 2018

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通过变异性研究确定大麻素CB1受体的正基调节器结合部位

Hayley M Green1, Daniel M J Fellner2, David B Finlay1

  • 1Department of Pharmacology and Toxicology, School of Biomedical Sciences, University of Otago, Dunedin 9016, New Zealand.

Pharmaceuticals (Basel, Switzerland)
|February 24, 2024
PubMed
概括

针对大麻素CB1受体 (CB1) 的正基调制剂 (PAM) 提供了治疗潜力. 这项研究确定了关键的残留物和结合部位,揭示了ZCZ011部位对CB1的全激应作用至关重要.

关键词:
大麻素CB1受体的受体.在GAT228中,GAT228是GAT228中的一个.在GAT229中,我们可以使用GAT229.的 ZCZ01111 的情况.一种全osteric 激动主义.通过全osteric 调制.绑定网站 绑定网站

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Published on: February 20, 2018

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An Assay for Quantifying Protein-RNA Binding in Bacteria07:02

An Assay for Quantifying Protein-RNA Binding in Bacteria

Published on: June 12, 2019

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