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新型 σ2R/TMEM97 配体的结构-亲和关系

Grant D Walby1, Qi Gu1, Hongfen Yang1

  • 1Department of Chemistry, The University of Texas at Austin, Austin, TX 78712, United States.

Bioorganic chemistry
|March 3, 2024
PubMed
概括

研究人员探索了新型的西格玛2受体 (σ2R) /跨膜蛋白97 (TMEM97) 调节器. 配体结构显著影响着对 σ2R/TMEM97 的结合亲和力和选择性,而不是对 σ1R.

关键词:
结合性亲缘关系是一种结合性亲缘关系.计算式对接方式西格玛2受体/跨膜蛋白 97 97结构-亲密关系-关系.异循环的合成

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