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4-氧二乙烯以多重向性联体的形式存在于胺H3受体和胆酶的受体中

Beata Michalska1, Marek Dzięgielewski1, Justyna Godyń2

  • 1Department of Synthesis and Technology of Drugs, Medical University of Lodz, Muszynskiego 1, 90-151 Lodz, Poland.

ACS chemical neuroscience
|March 5, 2024
PubMed
概括

研究人员开发了新的化合物,向组胺H3受体 (H3R),并抑制ACHE/BuChE酶. 化合物ADS031通过将H3R对抗与酶抑制相结合,显示出对阿尔茨海默病治疗的前景.

关键词:
乙烯基胆 Estrase 抑制剂的使用乙基胆酶抑制剂 乙基胆酶抑制剂组织胺H3受体的受体.多重准多个目标神经退行性疾病是一种神经退行性疾病.多种药理学 多种药理学

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