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Updated: Jul 1, 2025

A Microwave-Assisted Direct Heteroarylation of Ketones Using Transition Metal Catalysis
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快速获取具有完全替代α-碳的异环氨基胺的断开连接

Shouliang Yang1, Fen Wang1, Stephanie Scales1

  • 1Pfizer Oncology Medicinal Chemistry, San Diego, California 92121, United States.

The Journal of organic chemistry
|March 5, 2024
PubMed
概括

一个新的单步合成使得有价值的基氨基胺的产生成为可能. 这种方法有效地产生复杂的异环化合物用于药物发现,克服了以前的合成限制.

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