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Updated: Jul 1, 2025

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基于机制的血清蛋白酶宏循环抑制剂

Vishnu C Damalanka1, Victoria Banas1, Paolo De Bona1

  • 1Department of Biochemistry & Molecular Biophysics, Washington University School of Medicine, Saint Louis, Missouri 63110, United States.

Journal of medicinal chemistry
|March 13, 2024
PubMed
概括

新的宏环蛋白酶抑制剂克服了类药物限制. 这些化合物显示出更好的选择性,稳定性和药理动力学特性,为药物发现提供了一种新的策略.

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