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Updated: Jun 30, 2025

Synthesis and Structure Determination of µ-Conotoxin PIIIA Isomers with Different Disulfide Connectivities
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Published on: October 2, 2018

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含有稳定的碳化合物键的psilocybin类型的合成和生物活性

Marthe Vandevelde1, Andreas Simoens1, Bavo Vandekerckhove1

  • 1Department of Green Chemistry and Technology, Synthesis, Bioresources and Bioorganic Chemistry Research Group, Ghent University Coupure Links 653 9000 Ghent Belgium chris.stevens@ugent.be.

RSC medicinal chemistry
|March 22, 2024
PubMed
概括

合成了具有稳定的P-C键的新型psilocybin类似物. 这些化合物对5-HT2A和5-HT2B血清素受体表现出良好的结合亲和力,其中一个模拟物表现出对psilocin的增强5-HT2A选择性.

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