Marco Orleni1,2,3, Jan H Beumer4,5,6

  • 1Cancer Therapeutics Program, UPMC Hillman Cancer Center, Room G27E, Hillman Research Pavilion, 5117 Centre Avenue, Pittsburgh, PA, 15213-1863, USA.

概括

塔泽米托斯塔特是一种新的FDA批准的EZH2抑制剂,用于特定的癌症. 它通过阻断EZH2,一个关键蛋白质,并显示了有前途的结果在临床试验中,先进的上皮质肉瘤和卵泡淋巴瘤.

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