使3-oxetanyllithium使

Philipp Natho1, Marco Colella1, Michael Andresini1

  • 1FLAME-Lab, Flow Chemistry and Microreactor Technology Laboratory, Department of Pharmacy-Drug Sciences, University of Bari "A. Moro", Via E. Orabona 4, 70125, Bari, Italy.

Organic letters
|March 28, 2024
PubMed
概括

我们生成并使用不稳定的3-oxetanyllithium,一种新型核爱好者,用于合成候选药物. 这种方法通过使用氧乙环作为生物异体来改善药物特性.