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Updated: Jun 29, 2025

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在NSCLC中用于突变选择性和可逆第四代EGFR-TKI临床开发的化学支架

Emiliano Laudadio1, Luca Mangano2, Cristina Minnelli3

  • 1Department of Science and Engineering of Matter, Environment and Urban Planning, Marche Polytechnic University, 60131 Ancona, Italy.

ACS chemical biology
|March 29, 2024
PubMed
概括

新的EGFRTKI正在开发中,以对抗非小细胞肺癌 (NSCLC) 的耐药性. 本综述涵盖了针对EGFR突变的下一代药物,如T790M和C797S.

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