G蛋白结合受体 (GPCRs):结构,机制和药物发现方面的进展

Mingyang Zhang1,2, Ting Chen3, Xun Lu2

  • 1Key Laboratory of Protection, Development and Utilization of Medicinal Resources in Liupanshan Area, Ministry of Education, Peptide & Protein Drug Research Center, School of Pharmacy, Ningxia Medical University, Yinchuan, 750004, China.

概括

G蛋白结合受体 (GPCR) 是主要的药物标. 这项研究回顾了GPCR结构,药物相互作用和全性机制,指导了这种重要的受体家族的未来药物设计.

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