发现了针对HER2的新型胺 - - 坎プト素结合物的发现,该结合物具有选择性癌症治疗的有效抑制作用

Hanyu Wu1, Yunxiao Liu1, Jiaqi Zhou1

  • 1Centre of Drug Discovery, State Key Laboratory of Natural Medicines, China Pharmaceutical University, Nanjing 210009, China.

Bioorganic chemistry
|April 21, 2024
PubMed
概括

研究人员开发了用于向癌症治疗的新型类药物联合体 (PDC). 最佳化合物Z8显示出强大的抗瘤活性和对HER2阳性细胞的高生物安全性,提供了一个有前途的新策略.

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