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Updated: Jun 13, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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通过分子建模发现TAAR1激动性的新型化疗型

Giancarlo Grossi1, Naomi Scarano1, Francesca Musumeci1

  • 1Department of Pharmacy, Section of Medicinal Chemistry, School of Medical and Pharmaceutical Sciences, University of Genoa, Viale Benedetto XV, 3, 16132 Genoa, Italy.

Molecules (Basel, Switzerland)
|April 27, 2024
PubMed
概括

研究人员确定了新胺-胺醇化合物作为TAAR1 (Trace Amine Associated Receptor 1) 的有前途的激动剂. 这些发现推动了针对TAAR1.1的新治疗剂的开发.

关键词:
阿尔法折叠是什么意思在TAAR1中,TAAR1是TAAR1.激进分子的激进分子.分子对接的分子对接.微量氨基受体的微量氨基受体.

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