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Updated: Jun 27, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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对大麻素2受体的宏环调节剂的发现和开发

Nataša Tomašević1, Fabiola Susanna Emser1, Edin Muratspahić1

  • 1Center for Physiology and Pharmacology, Institute of Pharmacology, Medical University of Vienna, Vienna, Austria.

The Journal of biological chemistry
|April 28, 2024
PubMed
概括

研究人员发现了 vodo-C1,一种来自植物的循环,可以激活大麻素2型受体 (CB2R). 修改后的版本充当了对手,为CB2R药物开发提供了新的途径.

关键词:
与G蛋白结合受体的受体是G蛋白结合受体.一个全osteric调节器.大麻素2型受体受体2型受体这是一种类.植物植物植物植物植物.

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