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Updated: Jun 27, 2025

Yeast Luminometric and Xenopus Oocyte Electrophysiological Examinations of the Molecular Mechanosensitivity of TRPV4
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Published on: December 31, 2013

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不同激素的TRPV3激活伴随着从瓦尼洛伊德部位的脂质解离

Kirill D Nadezhdin1, Arthur Neuberger1, Lena S Khosrof1

  • 1Department of Biochemistry and Molecular Biophysics, Columbia University, New York, NY, USA.

Science advances
|May 1, 2024
PubMed
概括

结构揭示了四大麻 (THCV) 和2-aminoethoxydiphenylborane (2-APB) 如何激活TRPV3通道. 两种激动剂,尽管结合了不同的部位,但打开了道并取代了脂质,为TRPV3功能和药物设计提供了洞察力.

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