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Updated: Jun 27, 2025

A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

Published on: January 21, 2020

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与N-Arylcinnamylamines竞争的多米诺诺维纳吉尔循环序列

Mihály Kajtár1,2, Sándor Balázs Király1, Attila Bényei3

  • 1Department of Organic Chemistry, University of Debrecen, Debrecen 4002, Hungary.

The Journal of organic chemistry
|May 1, 2024
PubMed
概括

研究了N-arylcinnamylamines的Domino Knoevenagel循环反应,揭示了五种不同的循环路径. 从这些反应中获得的一些新型异环化合物表现出有前途的抗增殖活性.

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