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Updated: Jun 27, 2025

A Rapid and Quantitative Fluorimetric Method for Protein-Targeting Small Molecule Drug Screening
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A Rapid and Quantitative Fluorimetric Method for Protein-Targeting Small Molecule Drug Screening

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辐射非离子表面活性剂对药物蛋白结合的作用

E Paul Raj1, Puspalata Rajesh2,3, S Anjali1

  • 1Department of Chemistry, Annamalai University, Annamalai Nagar, India.

Journal of biomolecular structure & dynamics
|May 2, 2024
PubMed
概括

马辐射增强了药物与蛋白质的结合相互作用. 这项研究表明,像Pluronic F-127这样的辐射表面活性剂可以改善与药物ornidazole和telmisartan的结合 afinity 对牛血清白蛋白.

关键词:
在 BSA 系统系统中,马辐射辐射的作用分子性质的变化.药物与蛋白质结合的药物.分子对接的分子对接.

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