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Updated: Jun 26, 2025

Synthesis of Indoxyl-glycosides for Detection of Glycosidase Activities
09:10

Synthesis of Indoxyl-glycosides for Detection of Glycosidase Activities

Published on: May 27, 2015

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作为潜在的glyoxalase-I抑制剂的新型 antraquinone 胺基衍生物

Mohammed Al-Akeedi1, Manal Najdawi1, Qosay Al-Balas2

  • 1Department of Applied Pharmaceutical Sciences and Clinical Pharmacy, Faculty of Pharmacy, Isra University, Amman, Jordan.

Journal of medicine and life
|May 13, 2024
PubMed
概括

研究人员发现了新的 antraquinone 胺基衍生物,可以抑制 Glyoxalase-I (Glo-I),一种与癌症有关的酶. 化合物MQ3通过有效地阻断Glo-I活性,显示出作为抗癌剂的显著潜力.

关键词:
CDOCKER 是一个CDOCKER.甘氨酸-I 的含量.炭氨酸胺衍生物的甲基胺衍生物.分子对接的分子对接.分子动力学分子动力学药物动力学 药物动力学结合组 是一种结合组.

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