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Updated: Jun 26, 2025

Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines

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设计,合成和生物活性的三甲基替代甲醇衍生物的设计,合成和生物活性

Lefeng Dong1, Weiguo Wang1, Liqi Zhou2

  • 1Shanghai Key Laboratory of Chemical Biology, School of Pharmacy, East China University of Science and Technology, Shanghai 200237, China.

Journal of agricultural and food chemistry
|May 17, 2024
PubMed
概括

新的甲酸杀虫剂被合成,以减少毒性. 化合物8d对斑马鱼的毒性比fipronil低14倍,为害虫控制提供了更安全的替代品.

关键词:
杀虫活动 杀虫活动分子对接的分子对接.菲尼尔皮拉 (Phenylpyrazole) 是一种可怕的药物.对斑马鱼的毒性三甲基团是三甲基团的组成部分.

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