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Updated: Jun 25, 2025

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在新的14-基-6-oxomorphinans的enantioselective合成

Jonathan C Moore1,2, Louis Modell3, Jacqueline R Glenn4,5

  • 1The GlaxoSmithKline Carbon Neutral Laboratories for Sustainable Chemistry, University of Nottingham, Jubilee Campus, Triumph Road, Nottingham, NG7 2TU, UK. hon.lam@nottingham.ac.uk.

Chemical communications (Cambridge, England)
|May 24, 2024
PubMed
概括

开发了一种合成14-基-6-oxomorphinans的新方法. 这一途径成功地产生了4,5-desoxynaltrexone和4,5-desoxynaloxone,随后评估了它们的阿片类受体活性.

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