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尼克洛萨米德强化TMEM16A,并诱导血管收缩

Pengfei Liang1, Yui Chun S Wan1, Kuai Yu2

  • 1Department of Biochemistry, Duke University School of Medicine, Durham, NC, USA.

The Journal of general physiology
|May 30, 2024
PubMed
概括

尼克洛萨米德,以前认为可以抑制TMEM16A通道,实际上在生理条件下增强了它们. 这一发现表明,它在治疗喘和COPD等疾病时应该谨慎使用.

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