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Updated: Jun 24, 2025

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purin-5-N-isosteresas抗炎剂的合成,对接和生物评估

Ahmed M El-Saghier1, Souhaila S Enaili1,2, Aly Abdou1

  • 1Chemistry Department, Faculty of Science, Sohag University 282524 Sohag Egypt el.saghier@science.sohag.edu.eg.

RSC advances
|June 4, 2024
PubMed
概括

新合成的特里亚-特里亚衍生物通过抑制循环氧化酶 (COX) 酶表现出强大的抗炎作用. 这些化合物表现出与印米他辛相比更高的疗效,这表明有可能开发新的抗炎药物.

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