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Updated: Jun 24, 2025

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission

Published on: August 16, 2018

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结构-活性关系和功能评估大麻素类型-1受体

Shujie Wang1, Xinru Tian1, Suresh Paudel1

  • 1Pharmacology Laboratory, College of Pharmacy, Chonnam National University, Gwangju 61186, Republic of Korea.

Biomolecules & therapeutics
|June 6, 2024
PubMed
概括

研究人员确定了大麻素受体1 (CB1R) 配体的关键结构特征,以改善药物设计. 这项研究增强了对CB1R配体的理解,用于神经心理和神经退行性疾病的潜在治疗.

关键词:
大麻素1型受体受体1型受体埃尔克·埃尔克是什么意思这是一种G蛋白质蛋白质,G蛋白质蛋白质.连接物亲和力 连接物亲和力结构与活动的关系.

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