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Updated: Jun 24, 2025

Formulating and Characterizing an Exosome-based Dopamine Carrier System
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2- propyl-β-cyclodextrin 纳入复合体形成对多巴胺受体-配体相互作用的影响 - 一个案例研究

Lukas Zell1, Thomas S Hofer2, Mario Schubert3

  • 1Department of Pharmaceutical and Medicinal Chemistry, Institute of Pharmacy, Paracelsus Medical University, 5020 Salzburg, Austria; Research and Innovation Center for Novel Therapies and Regenerative Medicine, Austria.

Biochemical pharmacology
|June 7, 2024
PubMed
概括

环氧德克斯含复合物可以增强药物溶解性,但可能会改变体外结合亲和力. 这种依赖于连接体的效应意味着它们不能被普遍推用于改善药物发现研究中的可溶性.

关键词:
2 - 基基-β - 循环环德克斯特林.多巴胺受体的连接体是多巴胺受体.在状的中.在体外 (in vitro) 的情况下.包容性复杂的包容性复杂的半经验性的量子化学

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