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Updated: Jun 23, 2025

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纳瓦卡普兰特是一种新型和选择性的卡帕阿片类受体对抗剂,没有与阿片类药物相关的滥用相关的激素特性

Filomene G Morrison1, Lori Jean Van Orden1, Karla Zeitz1

  • 1Neumora Therapeutics, Inc., 490 Arsenal Way, Watertown, MA, 02472, USA.

Neuropharmacology
|June 14, 2024
PubMed
概括

纳瓦卡普兰特是一种选择性的卡帕阿片类受体 (KOR) 抗剂. 这项研究证实了其KOR抗性质和缺乏激素活性,表明它有可能在没有滥用责任的情况下治疗严重抑郁症.

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