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Updated: Jun 23, 2025

Protocol for the Synthesis of Ortho-trifluoromethoxylated Aniline Derivatives
08:43

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Published on: January 19, 2016

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快速电友性211 在三甲基米尔基的亚化时

Marius Müller1,2, Umberto Maria Battisti1, Merlin Zabrocki1

  • 1Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Universitetsparken 2, 2100, Copenhagen, Denmark.

ChemPlusChem
|June 14, 2024
PubMed
概括

新的三甲基基基使得能有效合成放射性标记的astatine-211 (211At) 化合物. 这种方法为富含电子和缺乏电子的基质提供了高放射化学转换,适合用于制药应用.

关键词:
阿斯类药物-211电友芳香替代的电友芳香替代放射性药物 放射性药物 放射性药物三酸酸三酸三酸三酸三酸三酸三酸三酸三甲基基尔米尔类.

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