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Updated: Jun 23, 2025

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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化学信息学 研究佐地亚泽-1,2,3-二醇衍生物的向布基胆酶

Yassine El Allouche1, Marwa Alaqarbeh2, Abdellah El Aissouq3

  • 1Laboratory of Processes, Materials, and Environment (LPME), Faculty of Science and Technology, Sidi Mohamed Ben Abdellah University, Fez, Morocco. yassine.elallouche@usmba.ac.ma.

Journal of fluorescence
|June 17, 2024
PubMed
概括

新设计的二-1,2,3-二醇衍生物显示出作为阿尔茨海默病的布基胆酶 (BuChE) 抑制剂的前景. 体内研究预测了有利的类似药物的特性和稳定的酶相互作用,为新疗法铺平了道路.

关键词:
接收人 接收人阿尔茨海默氏症是阿尔茨海默氏症的一种疾病.这是一种BuChE酶.分子对接是分子对接.分子动力学分子动力学在QSAR中使用QSAR.

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