应用三脚式尿素受体与抗瘤药物结合,康布列塔-A4酸盐

Yu Kong1, Rong Zhang1, Boyang Li2

  • 1Key Laboratory of Medicinal Molecule Science and Pharmaceutics Engineering, Ministry of Industry and Information Technology, School of Chemistry and Chemical Engineering, Beijing Institute of Technology, Beijing 102488, China.

PubMed
概括

研究人员开发了一种新型的六氨酸离子受体 (L),以改善酸盐药物,如Combretastatin-A4酸盐 (CA4P) 的传递. 这种受体通过键有效地结合CA4P,增强其用于药物递送应用的潜力.