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Updated: Jun 23, 2025

Homogeneous Time-resolved Förster Resonance Energy Transfer-based Assay for Detection of Insulin Secretion
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在老鼠肌管中发现了带有两个氨基功能的光环,作为SHIP2抑制剂,具有胰岛素敏感作用

Phei Ching Lim1, Beow Keat Yap1, Yi Juin Tay1

  • 1School of Pharmaceutical Sciences, Universiti Sains Malaysia Minden 11800 Penang Malaysia chongyew@usm.my +604 653 4086.

RSC medicinal chemistry
|June 24, 2024
PubMed
概括

新的奥龙化合物被开发为SHIP2的小分子抑制剂 (SH2域含有内醇5-酸酶2). 这些新型SHIP2抑制剂增强葡萄糖吸收,显示出作为口服胰岛素敏感剂的潜力.

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