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Updated: Jun 22, 2025

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维生素D受体对抗剂的结构和抗癌活性

Agnieszka Powała1, Teresa Żołek1, Geoffrey Brown2

  • 1Department of Organic and Physical Chemistry, Faculty of Pharmacy, Medical University of Warsaw, 1 Stefana Banacha, 02-097 Warsaw, Poland.

International journal of molecular sciences
|June 27, 2024
PubMed
概括

维生素D化合物被转化为活性激素,通过维生素D受体调节基因表达. 目前正在开发用于癌症治疗的类似药物,其血效应降低.

关键词:
在 VDR 带结合域中,VDR 带结合域酸醇是一种酸.维生素D是维生素D的重要组成部分.维生素D的抗癌类型类似物.维生素D的代谢物和类似物.维生素D受体 (VDR) 是一种维生素D受体.

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